Binding of the Dual-Action Anti-Parkinsonian Drug AG-0029 to Dopamine D2 and Histamine H3 Receptors: A PET Study in Healthy Rats

Nafiseh Ghazanfari
, Aren van Waarde
, Janine Doorduin
, Jürgen W. A. Sijbesma
, Maria Kominia
, Martin Koelewijn
, Khaled Attia
, David Vállez-García
, Antoon T.M. Willemsen
, André Heeres
, Rudi A. J. O. Dierckx
, Ton J. Visser
, Erik de Vries
, Philip H. Elsinga

Symeres
Rijksuniversiteit Groningen, Universitair Medisch Centrum Groningen, Afdeling Nucleaire Geneeskunde en Moleculaire Beeldvorming

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11 Article
1 Report
1 Poster
1 Patent

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2023
Substituted anilides from chitin-based 3-acetamido-furfural
van der Loo, C., Kaniraj, J. P., Wang, T., Pouwer, K., Broekman, O., Borst, M., Heeres, A., Deuss, P. & Minnaard, A., 5 okt. 2023, In: Organic and Biomolecular Chemistry. 21, 41, blz. 8372-8378 7 blz.
Onderzoeksoutput: Article › Academic › peer review

Open Access
2022
Advantages of Producing Aromatics from Propene over Ethene Using Zeolite-Based Catalysts
Butolia, P. S., Xi, X., Winkelman, J. G. M., Stuart, M. C. A., van Akker, M., Heeres, A., Heeres, H. J. & Xie, J., 11 okt. 2022, In: Chemie Ingenieur Technik - CIT. 94, 11, blz. 1845-1852 8 blz.
Onderzoeksoutput: Article › Academic › peer review

Open Access
A time- and space-resolved catalyst deactivation study on the conversion of glycerol to aromatics using H-ZSM-5
He, S., Goldhoorn, H. R., Tegudeer, Z., Chandel, A., Heeres, A., Stuart, M. C. A. & Heeres, H. J., 15 apr. 2022, In: Chemical Engineering Journal. 434, 134620.
Onderzoeksoutput: Article › Academic › peer review

Open Access
Pharmacokinetic Modeling of [11C]GSK-189254, PET Tracer Targeting H3 Receptors, in Rat Brain
Ghazanfari, N., van Waarde, A., Doorduin, J., Sijbesma, J. W. A., Kominia, M., Koelewijn, M., Attia, K., T.M. Willemsen, A., Visser, T. J., Heeres, A., Dierckx, R. A. J. O., de Vries, E. & Elsinga, P., 16 feb. 2022, In: Molecular Pharmaceutics. 19, 3, blz. 918–928 11 blz.
Onderzoeksoutput: Article › Academic › peer review

Open Access
Studying Telmisartan Plasma Exposure, Kidney Distribution, Receptor Occupancy, and Response in Patients With Type 2 Diabetes Using [11C]Telmisartan
van der Hoek, S., Mulder, D. J., T.M. Willemsen, A., Visser, T. J., Heeres, A., Slart, R. H. J. A., Elsinga, P. H., Heerspink, H. J. L. & Stevens, J., 7 sep. 2022, In: Clinical Pharmacology & Therapeutics. 112, 6, blz. 1264-1270 7 blz.
Onderzoeksoutput: Article › Academic › peer review

Open Access
2021
Catalytic Conversion of Free Fatty Acids to Bio-Based Aromatics: A Model Investigation Using Oleic Acid and an H-ZSM-5/Al2O3 Catalyst
He, S., Klein, F., Kramer, T. S., Chandel, A., Tegudeer, Z., Heeres, A. & Heeres, H. J., 10 jan. 2021, In: ACS Sustainable Chemistry and Engineering. 9, 3, blz. 1128-1141 14 blz.
Onderzoeksoutput: Article › Academic › peer review

Open Access
Catalytic conversion of glycerol and co-feeds (fatty acids, alcohols, and alkanes) to bio-based aromatics: remarkable and unprecedented synergetic effects on catalyst performance
He, S., Kramer, T. S., Sukmayanda Santosa, D., Heeres, A. & Heeres, H. J., 18 dec. 2021, In: Green Chemistry. 24, 2, blz. 941-949 9 blz.
Onderzoeksoutput: Article › Academic › peer review

Open Access
Catalytic conversion of glycerol to bio-based aromatics using H-ZSM-5 in combination with various binders
He, S., Goldhoorn, H. R., Tegudeer, Z., Chandel, A., Heeres, A., Liu, C., Pidko, E. & Heeres, H. J., okt. 2021, In: Fuel Processing Technology. 221, 106944.
Onderzoeksoutput: Article › Academic › peer review

Open Access
GMP Compliant Synthesis of [18F]Canagliflozin, a Novel PET Tracer for the Sodium−Glucose Cotransporter 2
van der Hoek, S., Antunes, I. F., Attia, K. A., Jacquet, O., Heeres, A., Bulthuis, M., Zijlma, R., Boersma, H. H., van Goor, H., Visser, T. J., Heerspink, H. J. L., Elsinga, P. H. & Stevens, J., 8 nov. 2021, In: Journal of Medicinal Chemistry. 64, 22, blz. 16641–16649 9 blz.
Onderzoeksoutput: Article › Academic › peer review

Open Access
GMP Compliant Synthesis of Canagliflozin, a Novel PET Tracer for the Sodium−Glucose Cotransporter 2
Heeres, A., van der Hoek, S., Antunes, I. F., Attia, K. A., Jacquet, O., Bulthuis, M., Zijlma, R., Boersma, H. H., van Goor, H., Visser, T. J., Heerspink, H. J. L., Elsinga, P. H. & Stevens, J., 8 nov. 2021, In: Journal of Medicinal Chemistry.
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2020

Catalytic conversion of pure glycerol over an un-modified H-ZSM-5 zeolite to bio-based aromatics
Heeres, A., He, S., Zuur , K., Sukmayanda Santosa, D., Liu, C., Pidko, E. & Heeres, H. J., sep. 2020, (E-pub ahead of print) In: Applied Catalysis B: Environment and Energy. 281, 14 blz.
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Binding of the Dual-Action Anti-Parkinsonian Drug AG-0029 to Dopamine D2 and Histamine H3 Receptors: A PET Study in Healthy Rats

Onderzoekersoutput

Zoekresultaten

2023

2022

2021

2020